Chemical CompoundsAZD4877

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M3672

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Description

AZD4877 is a specific, potent inhibitor of Eg5. AZD4877 selectively inhibits microtubule motor protein KSP (also called kinesin-5 or Eg5), which may result in the inhibition of mitotic spindle assembly. AZD4877 is generally well-tolerated with pharmacodynamic evidence of target inhibition in circulating PBMCs. AZD4877 was generally tolerable in patients with advanced urothelial cancer.

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