
BMS-740808
M3268
Brand
No Brand
Description
BMS-740808 is a highly potent, selective, efficacious, and orally bioavailable blood coagulation factor Xa inhibitor with a Ki of 30 pM. It has a rapid onset of inhibition (2.7 × 107 M−1 /s) in vitro, selective (>1000-fold over other proteases), efficacious in the AVShunt thrombosis model, and orally bioavailable inhibitor of blood coagulation factor Xa.
Application
Reactivity