Chemical CompoundsPFI-1

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HY-16586

10 mM * 1 mL in DMSO10 mg50 mg100 mg

Brand

MCE

Description

PFI-1 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM in a cell-free assay.

Molecular Formula: C16H17N3O4S
Molecular Weight: 347.39
Target: Epigenetic Reader Domain
Pathway: Epigenetics
Solubility: 10 mM in DMSO

Application

Reactivity

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